TTR

Chr 18AD

transthyretin

Also known as: AMYLD1, ATTR, CTS, CTS1, HEL111, HsT2651, PALB, TBPA

Transthyretin is a tetrameric carrier protein that transports thyroid hormones in plasma and cerebrospinal fluid and also transports retinol (vitamin A) by associating with retinol-binding protein. Mutations cause autosomal dominant hereditary transthyretin amyloidosis, which predominantly affects peripheral nerves and heart, as well as dystransthyretinemic hyperthyroxinemia and familial carpal tunnel syndrome. The gene shows moderate constraint against loss-of-function variants (LOEUF 0.763), and amyloidosis typically presents in adulthood with progressive polyneuropathy or cardiomyopathy.

OMIMResearchSummary from RefSeq, OMIM, UniProt
GOFmechanismADLOEUF 0.763 OMIM phenotypes
Clinical SummaryTTR
🧬
Gene-Disease Validity (ClinGen)
obsolete hereditary ATTR amyloidosis · ADDefinitive

Definitive — sufficient evidence for diagnostic panels

Population Constraint (gnomAD)
Moderately constrained gene (pLI 0.52) — some intolerance to loss-of-function variants.
💊
Clinical Trials
12 active or recruiting trials — potential therapeutic options may be available

Population Genetics & Constraint

gnomAD v4 — loss-of-function & missense intolerance

Moderate LoF intolerance
LoF Constraint
0.76LOEUF
pLI 0.516
Z-score 1.94
OE 0.16 (0.060.76)
Moderately constrained

Typical tolerance to LoF variation

Missense Constraint
1.01Z-score
OE missense 0.69 (0.550.86)
57 obs / 83.0 exp
Tolerant

Mild missense constraint

Observed / Expected Ratios
LoF OE0.16 (0.060.76)
00.351.4
Missense OE0.69 (0.550.86)
00.61.4
Synonymous OE0.90
01.21.6
LoF obs/exp: 1 / 6.2Missense obs/exp: 57 / 83.0Syn Z: 0.43
Curated Mechanism (G2P)Gene2Phenotype (DDG2P) ↗
definitiveTTR-related hereditary transthyretin (ATTR) amyloidosisGOFAD
DN
0.2598th %ile
GOF
0.4085th %ile
LOF
0.3163th %ile

The Badonyi & Marsh model scores gain-of-function highest, but genomic evidence most strongly supports loss-of-function (haploinsufficiency) as the primary mechanism.

LOF1 literature citation

Note: In-silico variant effect predictors (SIFT, PolyPhen, REVEL, CADD) may underestimate pathogenicity of missense variants in genes with GOF or DN mechanisms. Consider functional evidence and clinical context.

Literature Evidence

LOFResults showed that TTR haploinsufficiency (TTR+/-) leads to higher glucose in both plasma and in primary hepatocyte culture media and lower expression of the influx glucose transporters, GLUT1, GLUT3, and GLUT4.PMID:34199897

Predictions from Badonyi M, Marsh JA. PLoS ONE. 2024;19(8):e0307312.

ClinVar Variant Classifications

0 submitted variants in ClinVar

Protein Context — Lollipop Plot

TTR · protein map & ClinVar variants

Showing all ClinVar variants across the protein. Search a specific variant to highlight its position.

3D Protein StructureAlphaFold

Clinical Trials

Active and recruiting trials from ClinicalTrials.gov

MelanomaNon-Small-Cell Lung CancerThyroid Cancer

A Study to Learn About the Study Medicine Called PF-07799933 in People With Advanced Solid Tumors With BRAF Alterations.

RECRUITING
NCT05355701Phase PHASE1PfizerStarted 2022-07-05
PF-07799933binimetinibcetuximab
Malnutrition PregnancyMalnutrition in ChildrenMalnutrition (Calorie)

Early Life Malnutrition, Environmental Enteric Dysfunction and Microbiome Trajectories

RECRUITING
NCT07195006University of ZimbabweStarted 2025-01-27
Malnutrition in pregnancy as exposurePoor WASH living conditions as exposure
Cerebral Amyloid Angiopathy

SEarchiNg biomarkErs Cerebral Amyloid Angiopathy (SENECA)

RECRUITING
NCT04204642Fondazione I.R.C.C.S. Istituto Neurologico Carlo BestaStarted 2020-06-01
CAA patients data collection
Solid Tumor

A Study to Evaluate the Efficacy and Safety of TL118 in Solid Tumors Patients

RECRUITING
NCT06010342Phase PHASE2Teligene USStarted 2023-03-16
TL118 Capsule
Transthyretin Cardiac Amyloidosis

EFICAC-TTR Trial: Exercise and Nutritional Supplementation in Transthyretin Cardiac Amyloidosis

NOT YET RECRUITING
NCT07343999Phase NAUniversidad de BurgosStarted 2026-06
Usual CareHome-Based Multicomponent Exercise ProgramFiber Supplementation (Microcrystalline Cellulose)
Breast Cancer

Trial of Perioperative Endocrine Therapy - Individualising Care

ACTIVE NOT RECRUITING
NCT02338310Phase PHASE3Institute of Cancer Research, United KingdomStarted 2008-09
Aromatase Inhibitors
Advanced Solid TumorsHER2 Mutation

A Study to Learn More About How Well Treatment With Sevabertinib (BAY 2927088) Tablets Works and How Safe it is in Participants Who Have a Solid Tumor With Mutations of the Human Epidermal Growth Factor Receptor 2 (HER2)

RECRUITING
NCT06760819Phase PHASE2BayerStarted 2025-02-13
BAY2927088
Locally Advanced or Metastatic Solid TumorsLocally Advanced or Metastatic Non-small Cell Lung Cancer

A Study of XZP-5955 Tablets in Patients With NTRK or ROS1 Fusion Positive Locally Advanced or Metastatic Solid Tumors

RECRUITING
NCT04996121Phase PHASE1, PHASE2Xuanzhu Biopharmaceutical Co., Ltd.Started 2021-12-06
XZP-5955 tablets
Primary Central Nervous System Lymphoma

A Dose-escalating Pilot Study of Orelabrutinib for Newly-diagnosed PCNSL

ACTIVE NOT RECRUITING
NCT05036577Phase PHASE1Huashan HospitalStarted 2021-10-10
OrelabrutinibRituximabMethotrexate (MTX)
Advanced Mesenchymal Malignancies

Exploratory Clinical Study of TCR-T for MAGE-A4-positive Mesenchymal Malignancies

RECRUITING
NCT07467122Phase PHASE1Sun Yat-Sen Memorial Hospital of Sun Yat-Sen UniversityStarted 2026-03-15
TCR-T cells targeting MAGE-A4
ALL (Acute B-Lymphoblastic Leukemia)

A Clinical Study Exploring the Safety, Efficacy and Cell Metabolic Kinetics of Universal Car-t Cell Injection in CD19 and / or CD20 Positive Relapsed / Refractory B-cell Acute Lymphoblastic Leukemia in Adolescents, Children and Adults

RECRUITING
NCT07470073Phase EARLY_PHASE1Union Hospital, Tongji Medical College, Huazhong University of Science and TechnologyStarted 2026-04-01
CT1190B cell injection
Neoplasms

Study to Evaluate Safety and Antitumor Activity of Lete-Cel (GSK3377794) in HLA-A2+ Participants With NY-ESO-1 Positive Previously Treated Advanced (Metastatic or Unresectable) Synovial Sarcoma or Myxoid/Round Cell Liposarcoma

ACTIVE NOT RECRUITING
NCT06703346Phase PHASE2USWM CT, LLCStarted 2019-12-31
Letetresgene autoleucel (Lete-Cel (GSK3377794))CyclophosphamideFludarabine
Clinical Literature
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Full-Text Mentions
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