P2RX1

Chr 17

purinergic receptor P2X 1

Also known as: P2X1

The protein encoded by this gene belongs to the P2X family of G-protein-coupled receptors. These proteins can form homo-and heterotimers and function as ATP-gated ion channels and mediate rapid and selective permeability to cations. This protein is primarily localized to smooth muscle where binds ATP and mediates synaptic transmission between neurons and from neurons to smooth muscle and may being responsible for sympathetic vasoconstriction in small arteries, arterioles and vas deferens. Mouse studies suggest that this receptor is essential for normal male reproductive function. This protein may also be involved in promoting apoptosis. [provided by RefSeq, Jun 2013]

ResearchGenerating clinical summary…

Clinical highlights

Gene-disease validity (ClinGen)
inherited bleeding disorder, platelet-type · ADDisputedevidence questions this relationship
0
Active trials
17
Pubs (1 yr)
P/LP submissions
P/LP missense
1.21
LOEUF
Multiple*
Mechanism· predicted
Some data sources returned errors (1)

omim: Error: OMIM fetch failed: 429

Population Genetics & Constraint

gnomAD v4 — loss-of-function & missense intolerance

Tolerant — LoF & missense variants common in population
LoF Constraint?
1.21LOEUF
pLI 0.000
Z-score 0.81
OE 0.81 (0.561.21)
Tolerant

Highly tolerant — LoF variants common in population

Missense Constraint?
1.02Z-score
OE missense 0.81 (0.720.92)
197 obs / 241.7 exp
Tolerant

Mild missense constraint

Observed / Expected Ratios?
LoF OE?0.81 (0.561.21)
00.351.4
Missense OE?0.81 (0.720.92)
00.61.4
Synonymous OE?0.98
01.21.6
LoF obs/exp: 18 / 22.1Missense obs/exp: 197 / 241.7Syn Z: 0.14

ClinVar Variant Classifications

0 submitted variants in ClinVar

Protein Context — Lollipop Plot

P2RX1 · protein map & ClinVar variants

Showing all ClinVar variants across the protein. Search a specific variant to highlight its position.

Clinical Trials

Active and recruiting trials from ClinicalTrials.gov

No active trials found for this gene.

Search ClinicalTrials.gov →