GRK1

Chr 13

G protein-coupled receptor kinase 1

Also known as: GPRK1, RHOK, RK

The protein is a retina-specific kinase that phosphorylates rhodopsin to terminate phototransduction signaling, which is essential for scotopic vision and rapid adaptation to changes in illumination. Mutations cause Oguchi disease-2, a form of congenital stationary night blindness with autosomal recessive inheritance. The gene shows low constraint against loss-of-function variants, consistent with its recessive disease pattern.

OMIMResearchSummary from RefSeq, OMIM, UniProt
LOFmechanismLOEUF 0.821 OMIM phenotype
Clinical SummaryGRK1
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Gene-Disease Validity (ClinGen)
Oguchi disease · ARDefinitive

Definitive — sufficient evidence for diagnostic panels

Population Constraint (gnomAD)
Low constraint (pLI 0.00) — loss-of-function variants are relatively tolerated in the population.
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Clinical Trials
4 active or recruiting trials — potential therapeutic options may be available

Population Genetics & Constraint

gnomAD v4 — loss-of-function & missense intolerance

Tolerant — LoF & missense variants common in population
LoF Constraint
0.82LOEUF
pLI 0.000
Z-score 2.22
OE 0.49 (0.310.82)
Tolerant

Typical tolerance to LoF variation

Missense Constraint
0.43Z-score
OE missense 0.93 (0.851.02)
314 obs / 336.3 exp
Tolerant

Mild missense constraint

Observed / Expected Ratios
LoF OE0.49 (0.310.82)
00.351.4
Missense OE0.93 (0.851.02)
00.61.4
Synonymous OE0.97
01.21.6
LoF obs/exp: 11 / 22.3Missense obs/exp: 314 / 336.3Syn Z: 0.28
Curated Mechanism (G2P)Gene2Phenotype (DDG2P) ↗
definitiveGRK1-related Oguchi diseaseLOFAR

Predictions shown for reference only — model trained on dominant genes, not applicable to AR conditions.

DN
0.6455th %ile
GOF
0.74top 25%
LOF
0.2775th %ile

The Badonyi & Marsh prediction model was trained exclusively on dominant disease genes. Predictions are not reliable for genes with autosomal recessive inheritance and are shown at reduced opacity for reference only.

Predictions from Badonyi M, Marsh JA. PLoS ONE. 2024;19(8):e0307312.

ClinVar Variant Classifications

0 submitted variants in ClinVar

Protein Context — Lollipop Plot

GRK1 · protein map & ClinVar variants

Showing all ClinVar variants across the protein. Search a specific variant to highlight its position.

3D Protein StructureAlphaFold
Clinical Literature
Open Research Assistant →
Key Publications
Landmark & review papers · by relevance
PubMed
Top 5 results · since 2015Search PubMed ↗