GCH1

Chr 14ADAR

GTP cyclohydrolase 1

Also known as: DYT14, DYT5, DYT5a, GCH, GTP-CH-1, GTPCH1, HPABH4B

The protein is GTP cyclohydrolase I, the rate-limiting enzyme in tetrahydrobiopterin (BH4) biosynthesis that converts GTP to 7,8-dihydroneopterin triphosphate, with BH4 serving as an essential cofactor for aromatic amino acid hydroxylases and nitric oxide synthases. Loss-of-function mutations cause dopa-responsive dystonia (autosomal dominant) and BH4-deficient hyperphenylalaninemia (autosomal recessive). The pathogenic mechanism involves loss of enzyme function leading to BH4 deficiency and subsequent impairment of dopamine and other neurotransmitter synthesis.

OMIMResearchSummary from RefSeq, OMIM, UniProt, Mechanism
LOFmechanismAD/ARLOEUF 0.402 OMIM phenotypes
Clinical SummaryGCH1
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Gene-Disease Validity (ClinGen)
GTP cyclohydrolase I deficiency · SDDefinitive

Definitive — sufficient evidence for diagnostic panels

Population Constraint (gnomAD)
Highly constrained gene — heterozygous loss-of-function variants are very rare in the population (pLI 0.90). One damaged copy is likely sufficient to cause disease.
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Clinical Trials
3 active or recruiting trials — potential therapeutic options may be available

Population Genetics & Constraint

gnomAD v4 — loss-of-function & missense intolerance

LoF intolerant — likely haploinsufficient
LoF Constraint
0.40LOEUF
pLI 0.903
Z-score 2.93
OE 0.08 (0.030.40)
Highly constrained

More LoF-intolerant than ~75% of genes

Missense Constraint
1.52Z-score
OE missense 0.63 (0.530.76)
86 obs / 135.8 exp
Tolerant

Mild missense constraint

Observed / Expected Ratios
LoF OE0.08 (0.030.40)
00.351.4
Missense OE0.63 (0.530.76)
00.61.4
Synonymous OE1.16
01.21.6
LoF obs/exp: 1 / 11.9Missense obs/exp: 86 / 135.8Syn Z: -0.90
Curated Mechanism (G2P)Gene2Phenotype (DDG2P) ↗
definitiveGCH1-related dystoniaOTHERAD
definitiveGCH1-related GTP cyclohydrolase 1 deficiencyOTHERAR
DN
0.4686th %ile
GOF
0.3292th %ile
LOF
0.67top 25%

The highest-scoring mechanism for this gene is loss-of-function (haploinsufficiency).

LOFprediction above median · 1 literature citation · LOEUF 0.40

Literature Evidence

LOFStudy of a Swiss dopa-responsive dystonia family with a deletion in GCH1: redefining DYT14 as DYT5PMID:17804835

Predictions from Badonyi M, Marsh JA. PLoS ONE. 2024;19(8):e0307312. Mechanism ranking also informed by gnomAD constraint, ClinVar, and ClinGen data.

ClinVar Variant Classifications

0 submitted variants in ClinVar

Protein Context — Lollipop Plot

GCH1 · protein map & ClinVar variants

Showing all ClinVar variants across the protein. Search a specific variant to highlight its position.

3D Protein StructureAlphaFold
Clinical Literature
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