GALR1

Chr 18

galanin receptor 1

Also known as: GALNR, GALNR1

The GALR1 protein is a G-protein-coupled receptor for the neuropeptide galanin that inhibits adenylyl cyclase activity and is widely expressed in the brain, spinal cord, and peripheral tissues including small intestine and heart. Currently, no human diseases have been definitively associated with GALR1 mutations in the medical literature. The gene shows low constraint to loss-of-function variation (pLI = 0.0005, LOEUF = 1.347), suggesting that complete loss of function may be well tolerated.

Summary from RefSeq, UniProt
Research Assistant →
0
Active trials
20
Pubs (1 yr)
0
P/LP submissions
P/LP missense
1.35
LOEUF
Multiple*
Mechanism· predicted
Clinical SummaryGALR1
Population Constraint (gnomAD)
Low constraint (pLI 0.00) — loss-of-function variants are relatively tolerated in the population.

Population Genetics & Constraint

gnomAD v4 — loss-of-function & missense intolerance

Tolerant — LoF & missense variants common in population
LoF Constraint
1.35LOEUF
pLI 0.001
Z-score 0.86
OE 0.69 (0.371.35)
Tolerant

Highly tolerant — LoF variants common in population

Missense Constraint
-0.21Z-score
OE missense 1.04 (0.931.17)
209 obs / 200.7 exp
Tolerant

Tolerant to missense variation

Observed / Expected Ratios
LoF OE0.69 (0.371.35)
00.351.4
Missense OE1.04 (0.931.17)
00.61.4
Synonymous OE0.98
01.21.6
LoF obs/exp: 6 / 8.8Missense obs/exp: 209 / 200.7Syn Z: 0.17
DN
0.78top 25%
GOF
0.79top 25%
LOF
0.2387th %ile

This gene has evidence for multiple mechanisms of pathogenicity (gain-of-function and dominant-negative). Both the Badonyi & Marsh prediction and the broader genomic evidence point to gain-of-function as the predominant mechanism. Different variants in this gene may act through different mechanisms — interpret in context of the specific variant.

GOFprediction above median
DNprediction above median

Note: In-silico variant effect predictors (SIFT, PolyPhen, REVEL, CADD) may underestimate pathogenicity of missense variants in genes with GOF or DN mechanisms. Consider functional evidence and clinical context.

Predictions from Badonyi M, Marsh JA. PLoS ONE. 2024;19(8):e0307312.

ClinVar Variant Classifications

0 submitted variants in ClinVar

Protein Context — Lollipop Plot

GALR1 · protein map & ClinVar variants

Showing all ClinVar variants across the protein. Search a specific variant to highlight its position.

Clinical Trials

Active and recruiting trials from ClinicalTrials.gov

No active trials found for this gene.

Search ClinicalTrials.gov →
Clinical Literature
Open Research Assistant →